Vofopitant (GR205171) shi ne mai magani da abubuwa a matsayin wani NK 1 kamar tsoka mai amsa sigina ne antagonist . Yana da tasirin irin na antiemetic kamar yadda yake tare da sauran abokan adawar NK 1 kuma yana nuna ayyukan tashin hankali a cikin dabbobi. Anyi nazarin shi don aikace-aikace kamar jiyya ta phobia ta zamantakewa da rikicewar damuwa bayan tashin hankali, amma bai tabbatar da isasshen tasiri don siyarwa ba.

Vofopitant
type of chemical entity (en) Fassara
Bayanai
Ƙaramin ɓangare na chemical compound (en) Fassara
Sinadaran dabara C₂₁H₂₃F₃N₆O
Canonical SMILES (en) Fassara COC1=C(C=C(C=C1)N2C(=NN=N2)C(F)(F)F)CNC3CCCNC3C4=CC=CC=C4
Isomeric SMILES (en) Fassara COC1=C(C=C(C=C1)N2C(=NN=N2)C(F)(F)F)CN[C@H]3CCCN[C@H]3C4=CC=CC=C4
Ta jiki ma'amala da Tachykinin receptor 1 (en) Fassara
Subject has role (en) Fassara antiemetic (en) Fassara da NK1 receptor antagonists (en) Fassara

Duba kuma gyara sashe

  • NK 1 antagonist mai karɓa

Manazarta gyara sashe